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The main advantage of anastrozole as compared to antiestrogens (SERMs) such as tamoxifen or clomiphene consist in the fact that anastrozole blocks production of the aromatase enzyme, hence, prevents estradiol generation at the earliest stages, while antiestrogens only prevent contact of estradiol with the corresponding receptors by binding to them instead of estradiol, but don’t reduce its production in the body .Therefore, estradiol may still circulate in bloodstream in large amounts when you take antiestrogens. Anastrozole has no harsh side effects. Actually, affecting estradiol, it can suppress the level of the good cholesterol (HDL). However, when compared to AI like letrozole, anastrozole is preferable. Letrozole has quite a few side effects, the most common of which is erectile dysfunction. Although estradiol is known as a female hormone, men still need it. Estradiol maintains hormonal balance, participates in a great number of physiological processes and helps to gain muscle mass and strength.
Rus Bio Anastrozole History and Overview
Rus Bio - Anastrozole is an extremely powerful anti-estrogen officially belonging to the Aromatase Inhibitor (AI) family. Developed in the early 1990’s by Zenaca Pharmaceuticals and released in 1995 under the trade name Arimidex, this is perhaps the most commonly used AI and one of the most common anti-estrogens on the market. Arimidex has proven to be very effective in breast cancer treatment, even more so than traditional Nolvadex (Tamoxifen Citrate), and is a favorite anti-estrogen among many anabolic steroid users. Countless anabolic steroid users rely on Arimidex for on cycle estrogenic protection. Many anabolic steroids have the ability to aromatase and lead to excess estrogen, which in turn can lead to some of the most commonly associated side effects of anabolic steroid use.
Rus Bio Anastrozole Effects
As an anti-estrogen, Rus Bio - Anastrazole is valuable to the breast cancer patient as many forms of breast cancer feed off of the estrogen hormone. While perhaps an oversimplification, by administering Arimidex the effect starves the cancer. For decades Nolvadex was used for this purpose. Nolvadex has the ability to bind to the estrogen receptors, which in turn prevents estrogen from binding. However, AI’s like Arimidex actively inhibit the production of estrogen and reduce the actual amount of circulating hormone. In short, there is no estrogen available to cause damage to the breast cancer patient. In recent years, Rus Bio Anastrazole has become the leading anti-estrogen in the treatment of hormone receptor-positive breast cancer, especially among post-menopausal women. Once the cancer has subsided, it is not uncommon for Nolvadex to be introduced in order to keep the cancer at bay.
For the anabolic steroid user, the effects of Rus Bio Anastrazole are greatly appreciated in its ability to protect against estrogenic related side effects. Many anabolic steroids have the ability to promote estrogenic side effects due to the testosterone hormone’s interaction with the aromatase enzyme. As aromatization occurs, estrogen levels rise and this can lead to gynecomastia and excess water retention. When excess water retention becomes severe, this can also promote high blood pressure. Not all anabolic steroids aromatize, and as such, not all can lead to estrogenic related effects. However, many common steroids do carry the ability to promote estrogenic activity including Dianabol, all forms of Nandrolone and Boldenone to a degree and of course, all forms of testosterone heavily.
|Dosage||Men 0.5-1 mg/day|
|Active half-life||2 days|